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ANTI-DIABETIC DRUGS I. INSULIN I-A. SENSITIZERS 1. BIGUANIDES a. METFORMIN b. BUFORMIN c. PHENFORMIN 2. THIAZOLIDINEDIONES/PPAR a. PIOGLITAZONE b. RIVOGLITAZONE c. ROSIGLITAZONE d. TROGLITAZONE 3.

DUAL PPAR AGONISTS a. ALEGLITAZAR b. MURAGLITAZAR c. TESAGLITAZAR p1

I-B.SECRETAGOGUES 1.K+ATP a.SULFONYLUREAS aa.FIRST GENERATION SU (1) ACETOHEXAMIDE (2) CARBUTAMIDE (3) CHLORPROPAMIDE (4) TOLBUTAMIDE (5) TOLAZAMIDE (6) GLICLAZIDE bb.SECOND GENERATION SU (1) GLIBENCLAMIDE/GLYBURIDE (2) GLIPIZIDE (3) GLIQUIDONE (4) GLYCLOPYRAMIDE cc.THIRD GENERATION SU (1) GLIMEPIRIDE p2

1. K+ATP b. MEGLITINIDES/GLINIDES (1)NATEGLINIDE (2)REPAGLINIDE (3)MITIGLINIDE I-B.SECRETAGOGUES 2. GLP-1 ANALOGS a.EXENATIDE b.LIXISENATIDE c.LIRAGLUTIDE d.TASPOGLUTIDE e.ALBIGLUTIDE 3.DPP4 INHIBITORS(GLIPTIN) a.ALOGLIPTIN b.LINAGLIPTIN c.SITAGLIPTIN d.VILDAGLIPTIN e.SAXAGLIPTIN p3

I-C. ANALOGS/OTHER INSULINS 1. FAST ACTING INSULIN a. INSULIN ASPART(NOVOLOG) b. INSULIN LISPRO(HUMALOG) c. INSULIN GLULISINE(APIDRA) 2. SHORT ACTING INSULIN a. REGULAR INSULIN 3. INTERMEDIATE-ACTING INSULIN a. NPH 4. LONG ACTING INSULIN a. INSULIN GLARGINE(LANTUS) b. INSULIN DETEMIR(LEVEMIR) 5. ULTRA-LONG ACTING INSULIN a. INSULIN DEGLUDEC 6. INHALABLE INSULIN a. EXUBERA p4

II. OTHER ANTIDIABETIC DRUGS A. ALPHA-GLUCOSIDASE INHIBITORS 1. ACARBOSE 2. MIGLITOL 3. VOGLIBOSE B. AMYLIN ANALOG 1. PRAMLINTIDE C.SGLT2 INHIBITORS(-GLIFLOZIN) 1.SERGLIFLOZIN 2.REMOGLIFLOZIN 3.DAPAGLIFLOZIN 4.CANAGLIFLOZIN D. ALDOSE REDUCTASE INHIBITOR 1. TOLRESTAT

p5

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