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ADRENERGIC NERVOUS SYSTEM

ADRENOMIMETICS:
A: DIRECT ACTING
Non-Selective Selective
Adrenaline B1 B2 X1 X2
Noradrenaline Dobutamine Salbutamol General: Clonidine
Dopamine Dopexamine Terbutaline Phenylephrine Methyldopa
Bambuterol Methoxamine Guanabenze
Salmeterol Local:
Formoterol Imidazoline deriv:
Ritodrine Naphazoline
Isoxsuprine Xylometazoline
Oxymetazoline
Pseudoephidrine
ADRENOLYTICS:
Non-Selective Selective:
X: X1: X2:
i. 2-Haloalkylamines: ii. Ergot Alkyloids iii. Imidazolines Prazosin Yohimbine
Phenoxybenzamine Amine: Tolazoline Doxazosin
Ergotmetrine Phentolamine Terazosin
Methylergometrine Tamsulozin
Amino:
Ergotamine
Ergotoxine
Dihydroergotamine
Dihydroergotoxine
B:
Propranolol
Sotalol
Nadolol
Timolol
Pindolol
HISTAMINE/ANTIHISTAMINES
H1:
1st Generation:
1.Alkylamines 2. Ethanolamines 3. Ethyendiamines 4. Phenothiazines 5. Piperidines
Brompheniramine Diphenhydramine Trepelenamine Cyclizine Cyproheptadine
Chlorpheniramine Carbinoxamine Pyrilamine Meclizine
Dexchlorpheniramine Clemastine Buclizine
Doxylamine Hydroxyzine
2nd Generation:
Terfenadine
Fexofenadine
Asternizole
Loratidine
Desloratidine
Cetirizine
Azelastine
Mizolastine
Ebastine
Highly Sedative: Moderatly Sedative: Mild Sedative:
Promethazine Meclizine Cyclizine
Hydroxyzine Buclizine Clemastine
Diphenhydramine Cinnarizine Mepyramine
Dimenhydranate Cyproheptadine
Pheniramine
H2:
Cimetidine
Ranitidine
Fomotidine
Roxatidine
Loxatidine
SEROTONIN:
Agonists:
Buspirone Cisapride Sumatriptan LSD
Gepirone Renzapride
Ipsapirone
Antagonists:
Cyproheptadine Ketanserin Ondansetron Risperidone Clozapine
Methysergide Ritanserin Granisetron
Tropisetron
PROSTAGLANDINS:
Dinoprostone
Dinoprost
Carboprost
Misoprostol
Rioprostol
Enprostol
Alprostadil
Epoprostenol
Iloprost
NSAID's
Salicylates: Pyrazoline Deriv: Indole Deriv: Arylaliphatic Acids:
Aspirin Aminophenazone Indomethacin Acetic Acids: Proprionic Acids:
Diflunisal Metamizole Sulindac Diclofenac Ibuprofen
Methyl Salicylate Propiphenazone Tolmetin Ketodolac
Phenylbutazone Etodolac
Oxyphenbutazone
Fenamates: Pref COX2 Inhib: Selective COX2 Inhib:
Flufenamic Acid Ketorolac: Nimesulide Celecoxib
Mephanamic Acid Nefopam: Meloxicam Rofecoxib
Meclophenamic Acid Nabumetone Valdecoxib
B: INDIRECT ACTING C:MIXED ACTION
Amphetamines Ephidrine
Anorectic drugs: Metaraminol
Noradrenergic:
Phentermine
Phenylpropanolamine
Mazindol
Serotonergic:
Fenfluramine
Dexfenfluramine
Noradrenergic/Serotonergic:
Sibutramine
B: X&B:
Metoprolol Labetalol
Atenolol Carvedilol
Acebutalol Nebivolol
Bisoprolol Celiprolol
Esmolol
Celiprolol
P-Amino Phenol Deriv:
Phenacetine
Paracetamol
GENERAL ANESTHETICS:
1. INHALATION: 2.IV:
A: GASES B: VOLATILE LIQUIDS A: BARBITURATES B: BENZODIAZEPINES
Nitrous Oxide Halothane Secobarbital Diazepam
Cyclopropane Enflurane Methohexitone Na Lorazepam
Isoflurane Thiopentone Na Midazolam
Desflurane
Sevoflurane Propofol
Diethyl-Ether Ketamine
LOCAL ANESTHETICS:
1. ESTERS 2.AMIDES
Cocaine Lignocaine(Eutectic)
Procaine Prilocaine(Eutectic)
Tetracaine Ropivacaine
Chlorprocaine Etidocaine
Benzocaine Bupivacaine
Dibucaine
Mepivacaine
1. INJECTABLE 2.SURFACE
Low potency Interm potency High potency Soluble
Procaine Lignocaine Tetracaine cocaine
Chlorprocaine Prilocaine Bupivacaine lignocaine
Ropivacaine Tetracaine
Dibucaine Benoxinate
Insoluble
Benzocaine
Oxethazaine
HYPNOTICS:
1.BARBITURATES
Barbituric Acid
Long Acting: Intermed Acting: Short Acting: Ultra Short Acting:
Phenobarbitone Amobarbitol Butobarbitone Thiopentone
Mephobarbitone Secobarbitone Methohexitone
Pentobarbitone Hexobarbitone
2. BENZODIAZEPINES
Long Acting: Short Acting
Flurazepam Temazepam
Diazepam Traizolam
Nitrazepam Midazolam
Flunitazepam
3.NON-BENZODIAZEPINE
Zopiclone
Zolpidem
Zaleplon
C: OPIOIDS
Fentanyl
Morphine
Pethidine
ANTI-PARKINSON
1. DOPERMINERGIC SYSTEM 2. CHOLINERGIC SYSTEM
A: DOPAMINE PRECURSORS: A: CENTRAL ANTI-CHOL
Levodopa Trihexphenidyl
B: PERIPH DECARBOXYLASE INHIB: B: ANTI-HIST
Carbidopa
Benserazide
C: DOPAMINERGIC AGONISTS:
Bromocriptine
Pergolide
Piribenil
Ropinirole
Pramipexole
D: MOAb INHIB
Selegiline
E: COMT INHIB
Entacapone
Tolcapone
F: DOPAMINE FACILITATORS
Amantadine
ANTI-EPILEPTIC
1. BARBITURATES: 7. BENZODIAZEPINES:
Phenobarbitone Clonazepam
2. DEOXY-BARBITURATES: Diazepam
Primidone Clobazepam
3. HYDANTOINS: Lorazepam
Phenytoin 8. PHENYLTRIAZINE
4. IMINOSTILBENES: Lamotrigine
Carbamezapine 9. CYCLIC-GABA-ANALOGUE:
5. SUCCINAMIDES: Gabapentin
Ethosuxamide 10. NEW DRUGS
Mesuxamide Vigabatrine
Phensuxamide Tiagabine
6. ALYPHATIC CARB ACID Levetiracetam
Valproic Acid 11. OTHERS:
Topiramate
PSYCHOSTIMULANTS
METHYLXANTHINES:
Caffeine
Theophilline
Theobromine
OPIOID ANALGESICS/ANTAGONISTS
AGONISTS:
1. Natural 2. Semi-Synth 3. Synthetic
Morphine Heroin Pethidine
Codeine Hydromorphine Fentanyl
Thebaine Oxymorphine Alfentanyl
Papaverine Oxycodone Sulfentanyl
Noscapine Hydrocodone Remifentanyl
Methadone
Dextropropoxyphene
Tramadol
WEAK AGONISTS:
Buprenorphine
AGONIST/ANTAG:
Nalorphine
Pentazocine
Nalbuphine
Butorphanol
PURE ANTAG:
Naloxone
Naltrexone
Nalmefene
MENTAL ILLNESS:
1. ANTI-PSYCHOTIC
A:Phenothiazines B: Butyrophenones C: Thioxanthenes D: Heterocycles
Aliphatic side chains Haloperidol Thiothixene Pimozide
Chlorpromazine Trifluperidol Flupenthixol Loxapine
Levomepromazine Droperidol Reserpine
Triflupromazine Penfluridol
Pipiridine side chains
Thioridazine
Piperazine side chains
Trifluoperazine
Fluphenazine
2. ANTI-ANXIETY
A: Benzodiazepines B: Azapirones C: Anti-H D: B-Blockers
Diazepam Buspirone Hydroxyzine Propranolol
Oxazepam Gepirone
Lorazepam Ispapirone
Alprazolam
Chlordiazepoxide
Clonazepam
Nitrazepam
Flurazepam
3. ANTI-DEPRESSANTS
A: Reversible inhib of MOA B: Tricyclic C: Selective 5-HT Reuptake Inhib
MAOa NA,5-HT reuptake inhib Fluoxetine
Moclobemide Imipramine Fluvoxemine
Clorgyline Amitryptiline Paroxetine
MAOb Trimipramine Sertraline
Selegiline Doxapine Citalopram
MAO Clormipramine
Tranylcypromine NA reuptake Inhib
Phenelzine Desipramine
Nortryptalline
Amoxapine
MANIA:
Lithium
E: Indole deriv: F: New
Ziprasidon Olanzapine
Clozapine
Risperidone
Quetiapine
D: Atypical
Trazodone
Mianserin
Tianeptine
Amineptine
Venlafaxine
Mirtazapine
Bupropion
CARDIO GLYCOSIDES AND CONGESTIVE HEART FAILURE
Cardiac Glycosides Inotropic drugs
Digitoxin Doutamine
Digoxin Dopamine
Gitoxin Amrinone
Gitalin Milrinone
Strophantin-K
Strophantin-G
Convallotoxin
Acetyl-Digoxin
Acetyl-Strphanthidin
Deacetyl-Lanatoside
ANTI-ANGINAL/ANTI ISCHEMIC DRUGS
A: NITRATES B: B-BLOCKERS C: CALCIUM CHANNEL BLOCKERS D: K+ CH OPENERS E: OTHERS
Short Acting Propranolol Verapimil Diltiazem Nifedipine Prenylamine Nicorandil Dipyridamole
Glyceral trinitrate(nitroglyc) Nadolol Gallopamil Fostedil Nicardipine Fendiline Trimetazidine
Isosorbide Dinitrate Metoprolol Thiapamil Nictiazem Nimodipine Cinnarazine
Long Acting Anipamil Nisoldipine Flunarizine
Isosorbide Dinitrate Emopamil Felodipine
Isosorbide Mononitrate Ronipamil Isrudipine
Erythrityl Tetranitrate Niludipine
Penta Erythritil Tetranitrate Amlodipine
Molsidomine
HYPERTENSION
A: SYMPATHETIC NS B: VASODILATORS C: Ca CHANNEL BLOCKERS D: DIURETICS E: ACE-I
Central: Minoxidal Nifedipine Diltiazem Verapamil Thiazides: Enalapril
Methyldopa Nitroprusside Na Nitrendipine Mibefradil Benzothiazide Captoprl
Clonidine Diazoxide Amlodipine Chlorthiazide Ramipril
Guanabenz Hydralazines: Nicardipine Hydrochlorthiazide AT-II-Inhib
Guanfacine Hydralazines Isradipine Sulfonamides: Sartans
Ganglioplegics: Dihydralazine Indapamide
Trimethaphan Chlortalidone
X1-Blockers Metolazone
Prazosin Loop:
Terazosin Furosamide
Doxazosin K-Sparing
Trimazosin Spiranolactone
Indoramin
Urapidil
Ketanserin
B-Blockers X & B-Blockers
Non-Selective Selective Labetalol
Propranolol Acebutalol Celiprolol
Oxprenolol Atanolol Dilevalol
Pindolol Bisoprolol Nebivolol
Sotalol Metoprolol
Timolol Betaxolol
Nadolol
CARDIAC ARRHYTHMIAS
A: Na-Ch-Blockers B: B-Blockers C: Prolong Action Potential(K-blockers_ D: Ca-Ch-Blockers
IA: Propranolol Amiodarone Verapamil
Quinidine Diltiazem
Procainamide
Disopyramide
IB:
Lidocaine
Mexyletine
Phenytoin
IC:
Flecainide
Encainide
Lorcainide
Propafenone
DIURETICS
A: Loop B: Thiazide C: CA-Inhib D: K-Sparing E: Osmotic
Furosemide Chlorthiazide Acetazolamide Aldosterone Antag: Mannitol
Bumetanide Clorthalidone Spiranolactone Glycerin
Ethacrynic Acid Xipamide Epith Na-ch-Inhib Isosorbid
Indapamide Triamterene Urea
Clopamide Amiloride
COAGULATION DISORDERS
A: Anti-Coagulants B: Thrombolytics C: Anti-Platelet
Heparin Oral Streptokinase Aspirin
Low Molec Weight Heparins: Warfarin Urokinase Dipridamole
Enoxaparin Dicoumarol Alteplase Ticlopidine
Reviparin Acenocoumarol Anti-Thrombolytics Clopidogrel
Nadroparin Phenindione Epsilon amino-caproic acid Glycoprotein
Dalteparin Tranexamic Acid Abciximab
Haparinoids Aprotinin
Heparan Sulfate
Danaparoid
Lepirudin
Heparin Antag
Protamine Sulphate
PEPTIC ULCER
A: Dec Gastric Acid Sec B: Antacids C: Ulcer Protec D: Ulcer Healing E: Anti-Helico Bacter Pylori
Anti-H2 Sodium Bicarb Sucralfate Carbenoxolone Na Clarithromycin
Cimetidine Magnesium Hydrox Bismuth Amoxicillin+Omeprazole
Famotidine Magnesium Trisilicate Tetracylclin+Metronidazole
Ranitidine Aluminium Hydroxide Gel Tinidazol+Bismuth
Nizatidine Ca Carbonate Amox+Metro+Ranitidine
Loxatidine Amox+Clar+lansoprazol
Roxatidine
Proton-Pump Inhib
Omeprazole
Pantoprazole
Rabeprazole
Lansoprazole
Esomeprazole
Anti-Cholinerg
Atropine
Pirenzepine
Propantheline
PG Analogues
Misoprostol
Anti-Gastrin
Proglumide
CA-Inhib
Acetazolamide
BRONCHIAL ASTHMA
A: Bronchodilators B: Leukotriene Antag C: Mast Cell Stabilizers D: Corticosteroids
Sympathomimetics Montelukast Na Chromoglycate Beclomethasone diproprionate
Non-Selective Selective-B2 Zafirlukast Nedocromal Na Budenoside
Adrenaline Salbutamol Ketotifen Fluticasone proprionate
Ephedrine Terbutaline Flunisolide
Isoprenaline Bambuterol
Salmetarol
Formoterol
Methylxanthines
Caffeine
Theophyilline
Theobromine
Anti-Cholinergics
Ipratopium
Tiotropium

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