DRUGS
medpgnotes
Contents
ANTICHOLINESTERASE .................................................................................................................................................................................................................................. 2
AUTACOIDS .......................................................................................................................................................................................................................................................... 2
BETA BLOCKERS ................................................................................................................................................................................................................................................ 2
BISPHOSPHONATES ......................................................................................................................................................................................................................................... 2
CATARACT NUGGETS....................................................................................................................................................................................................................................... 3
CONDITION AND SPECIFIC DRUG ............................................................................................................................................................................................................... 4
CONDITION AND SPECIFIC SURGERY ....................................................................................................................................................................................................... 5
DIABETES NUGGETS ........................................................................................................................................................................................................................................ 6
DIFFERENT USAGE OF DRUGS ..................................................................................................................................................................................................................... 7
DRUG OF CHOICE ............................................................................................................................................................................................................................................... 7
DRUG KINETICS............................................................................................................................................................................................................................................... 11
FEW DRUG INTERACTIONS ........................................................................................................................................................................................................................ 11
MECHANISM OF ACTION OF DRUGS ....................................................................................................................................................................................................... 12
MONOCLONAL ANTIBODIES ...................................................................................................................................................................................................................... 19
NITRATES NUGGET ....................................................................................................................................................................................................................................... 19
OPIOID NUGGET .............................................................................................................................................................................................................................................. 20
PRODRUGS ........................................................................................................................................................................................................................................................ 20
SAFEST DRUGS IN PREGNANCY NUGGET............................................................................................................................................................................................. 21
STEROID DRUGS ............................................................................................................................................................................................................................................. 21
TREATMENT OF CHOICE ............................................................................................................................................................................................................................. 22
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ANTICHOLINESTERASE
ANTICHOLINESTERASE
Naturally occurring Anticholinesterase
Lipid Soluble Anticholinesterase
Blood brain barrier crossing Anticholinesterase
Anticholinesterase used in Myasthenia Gravis
Anticholinesterase used for Diagnosis of Mtasthenia
Gravis
Anticancer showing Anticholinesterase Property
Physostigmine
Neostigmine/Pyridostigmine
Edrophonium
Irinotecan
AUTACOIDS
FUNCTION
Most Important chemical elevating Hypothalamic
setpoint
Vasoconstrictor
Prostaglandins causing Renal Vasodilataion
Vasodilatation in blood vessels
Platelet Aggregation
Inhibition of Platelet aggregation
Chemotactic
Bronchoconstrictor
Slow reacting substance of anaphylaxis(SRSA)
AUTAOIDS
PGE2
PGF2
PGI2,PGE2
PGI2,PGE2,PGF2
TXA2
PGI2
LTB4
LTC4
LTD4
LTE4
BETA BLOCKERS
Most Cardioselective
Vasodilator Property
K+ Blocking Property
K+ Opening Property
Selective 2 blocker
Non Catecholamine acting selectively on
Nebivolol
Sotalol
Tilsolol
Butoxamine
Prenalterenol
BISPHOSPHONATES
st
1 Bisphosphonate Approved
Treatment of Postmenopausal Osteoporosis
Prevention of Steroid Induced Osteoporosis
Unique Administration Technique
Once Yearly i.v/Once Monthly Oral
Most Potent Drug for Treatment & Prevention of
Osteoporosis
Etindronate
Alendronate
Risendronate
Risendronate
Zolendronate
Idandronate
Bisphosphonates
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CATARACT NUGGETS
CATARACT NUGGETS
Anterior Polar
Anterior Capsular
Anterior Subscapular
Posterior Polar
Posterior Capsular
Posterior Subcapsular
Cataract
Cataract
Keratomalacia
Age Related
Punctate cataract
Visual Impairment/Cataract
Lamellar/Zonular cataract
Complicated Cataract with Posterior Capsular Opacities
Nuclear Cataract
Diabetic Cataract
Phacomorphic Glaucoma
Phacolytic Glaucoma
Subluxation/Dislocation of Lens
Phacoanaphylactic Uveitis
Galactitiol
Sorbitol
Oil Drop Cataract
Cataract
Steroid
SPECIFIC CATARACT
Snow Flake Cataract
Sunflower Cataract
Diabetes Mellitus
Wilsons disease
Chalcosis
Penetrating trauma
Blunt Trauma
Myotonica Dystrophica
Galactosemia
Hypermature Senile Cataract
Complicated Cataract
Ultraviolet
Infrared
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