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1

Diphenoxylate

:






.




2,5

0,025


1 2 4 8 40

5 10 4
48

: .
4-2
) 2.5 ( 3 ) (
9-4
5 3
9-12
4 5
12-16
2 3 10
12-18
4 2 6
2 4 ) 6 (
20 10 4

0.3 0.4 4
48



Blood Brain Barrier



)
(


) 1 :
25 (




.


.

) (Diphenoxylate
6 - 1 .



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,

, , , ,, , , ,
, , ,

CYP450
:

49 14 , , 2
14-12
:

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