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High protein binding Low protein High bio

Acetazolamide Amiloride Acetazolamide


Amiodarone Atenolol Aminophylline
Amitriptyline Carbimazole Carbamazepine
Aprepitant Cimetidine Ciprofloxacin
Aspirin Clonidine Clonidine
Azoles (ketoconazole, micoconzole Codeine Cyclizine
Bupivacaine Digoxin Diazoxide
Celecoxib Gabapentin Disopyramide
Cocaine Guanethidine Etoricoxib
Dantrolene Ketamine Flecainide
Diazepam Levetiracetam Isosorbide mononitrate
Diazoxide Metformin Lamotrigine
Diclofenac Methyldopa Levetiracetam
Droperidol Metoprolol Meloxicam
Etoricoxib Minoxidil Methadone
Fentanyl Morphine Metronidazole
Furosemide Neostigmine Mexiletine
Gliclazide Nicorandil Minoxidil
Hydralazine Paracetamol Oxycodone
Ibuprofen Pregabalin Paracetamol
Lorazepam Ranitidine Phenytoin
Losartan Salbutamol Pregabalin
Meloxicam Sotalol Procainamide
Methadone Tapentadol Quinidine
Midazolam Sotalol
Nifedipine Tenoxicam
Phenytoin
Prazosin
Propafenone
Propanolol
Propofol
Quinidine
Repaglinide
Ropivacaine
Sildenafil
Sodium valproate
Spironolactone
Tenoxicam
Thiopental
Thyroxine
Verapamil
Warfarin
Low bio Solely urine Bile excretion
Acebutolol Acetazolamide Azoles (ketoconazole, micoconzole
Acyclovir Atenolol Bosentan
Chlorpromazine Diazoxide Dipyridamole
Diamorphine Digoxin Pancuronium
Edrophonium Furosemide Phenytoin
Enoximone Gabapentin Prazosin
Etomidate Gelatins Rifampicin
Fentanyl Gentamicin Rocuronium
Flumazenil Gliclazide Vecuronium
Glycopyrollate Glycopyrollate
GTN Metformin
Isoprenaline Milrinone
Labetalol Omeprazole
Losartan Pregabalin
Methyldopa Pyridostigmine
Midazolam Sotalol
Morphine Sugammadex
Neostigmine Temazepam
Phenoxybenzamine Vigabatrin
Phentolamine
Propanolol
Propofol
Remifentanyl
Sildenafil
Tapentadol
Thiopental
Verapamil
P-Amiloride
pATENOLOLu

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