Memblok reseptor
Antihistamin
1st Generation
otonom
H1-receptor antagonist
2nd Generation
Menurunkan distribusi ke
Less lipid soluble than 1st CNS
generation
Ranitidine
H2
Antagonis
Famotidine
Nizatidine
H2
Antagonis Eliminasi dari tubuh melalui
metabolisme hepatic, glomerular
filtrasi & sekresi renal tubular