- Maraviroc (di CCR5) - Enfuvirtide (di gp41) Nucleoside analogues (NARTIs) - Efavirenz (EFV) - Lopinavir (LPV) - Raltegravir - Bevirimat
- Vicriviroc (di CCR5) - Zidovudine (ZDV/AZT) - Nevirapine (NVP) - Ritonavir (RTV/ r) - Elvitegravir - Elvucitabine
- Ibalizumab (di CD4) - Lamivudine (3TC) - Delavirdine - Nelvinafir
- Didanosine (ddi) - Lersivine - Saquinavir (SGV)
- Abacavir (ABC) - Etravirine - Amprenavir (APV)
- Emtricitabine (FTC) - Rilpivirin (RVP) - Atazanavir (ATV)
Nucleotide analogues (NtRTIs) - Darunavir (DRV)
- Tenofovir (TDV)